Daan van der Es
Universitair hoofddocent
- Naam
- Dr. D. van der Es
- Telefoon
- 071 5274513
- d.van.der.es@lacdr.leidenuniv.nl
- ORCID iD
- 0000-0003-3662-8177
Universitair hoofddocent
- Wiskunde en Natuurwetenschappen
- Leiden Academic Centre for Drug Research
- LACDR/Medicinal Chemistry
- Beerkens B.L.H., Andrianopoulou V., Wang X., Liu R., Westen G.J. P. van, Jespers W., IJzerman A.P., Heitman L.H. & Es D. van der (2024), N-Acyl-N-alkyl sulfonamide probes for ligand-directed covalent labeling of GPCRs: the adenosine A2B receptor as case study, ACS Chemical Biology 19(7): 1554-1562.
- Hollander L.S. den, Beerkens B.L.H., Dekkers S., Veldhoven J.P.D. van, Ortiz Zacarías N.V., Horst C. van der, Sieders E.G., Valk B. de, Wang J., IJzerman A.P., Es D. van der & Heitman L.H. (2024), Labeling of CC chemokine receptor 2 with a versatile intracellular allosteric probe, ACS Chemical Biology 19(9): 2070-2080.
- Beerkens B.L.H., Snijders I.M., Snoeck J., Liu R., Tool A.T.J., Le Dévédec S.E., Jespers W., Kuijpers T.W., Westen G.J.P. van, Heitman L.H., IJzerman A.P. & Es D. van der (2023), Development of an affinity-based probe to profile endogenous human adenosine A3 receptor expression, Journal of Medicinal Chemistry 66(16): 11399-11413.
- Beerkens B.L.H., Wang X., Avgeropoulou M., Adistia L.N., Veldhoven J.P.D. van, Jespers W., Liu R., Heitman L.H., IJzerman A.P. & Es D. van der (2022), Development of subtype-selective covalent ligands for the adenosine A2B receptor by tuning the reactive group, RSC Medicinal Chemistry 13(7): 850-856.
- Beerkens B.L.H., Koc C., Liu R., Florea B.I., Le Dévédec S.E., Heitman L.H., IJzerman A.P. & Es D. van der (2022), A chemical biological approach to study G protein-coupled receptors: labeling the adenosine A1 receptor using an electrophilic covalent probe, ACS Chemical Biology 17(11): 3131-3139.
- Yang X., Heitman L.H., IJzerman A.P. & Es D. van der (2021), Molecular probes for the human adenosine receptors, Purinergic Signalling 17: 85-108.
- Amelia T., Veldhoven J.P.D. van, Falsini M., Liu R., Heitman L.H., Westen G.J.P. van, Segala E., Verdon G., Cheng R.K.Y., Cooke R.M., Es D. van der & IJzerman A.P. (2021), Crystal structure and subsequent ligand design of a nonriboside partial agonist bound to the adenosine A2A receptor, Journal of Medicinal Chemistry 64(7): 3827-3842.
- Ortiz Zacarías N.V., Chahal K.K., Šimková T., Horst C. van der, Zheng Y., Inoue A., Theunissen E., Mallee L., Es D. van der, Louvel J., IJzerman A.P., Handel T.M., Kufareva I. & Heitman L.H. (2021), Design and characterization of an intracellular covalent ligand for CC chemokine receptor 2, Journal of Medicinal Chemistry 64(5): 2608-2621.
- Berni F., Kalfopoulou E., Gimeno Cardells A.M., Carboni F., Es D. van der, Romero-Saavedra F., Laverde D., Miklic K., Malic S., Rovis T.L., Jonjic S., Ali S., Overkleeft H.S., Hokke C.H., Diepen A. van, Adamo R., Jiménez-Barbero J., Marel G.A. van der, Huebner J. & Codée J.D.C. (2021), Epitope recognition of a monoclonal antibody raised against a synthetic glycerol phosphate based teichoic acid, ACS Chemical Biology 16(8): 1344-1349.
- Mever M. van, Willacey C.C.W., Zhang W., Drouin N.F.P., Christina A.E., Lindenburg P.W., Veldhoven J.P. D. van, Es D. van der, Harms A.C., Hankemeier T. & Ramautar R. (2021), Profiling acidic metabolites by capillary electrophoresis‐mass spectrometry in low numbers of mammalian cells using a novel chemical derivatization approach, Analytical Science Advances 3(1-2): 3-13.
- Enotarpi J.Tontini M. Balocchi C. Es D. van der Auberger L. Balducci E. Carboni F. Proietti D. Casini D. Filippov D.V. Overkleeft H.S. Marel G.A. van der Colombo C. Romano M.R. Berti F. Costantino P. Codeé J.D.C. Lay L. Adamo R. (2020), A stabilized glycomimetic conjugate vaccine inducing protective antibodies against Neisseria meningitidis serogroup A, Nature Communications 11: 4434.
- Yang X. Dilweg M.A. Osemwengie D. Burggraaff L. Es D. van der Heitman L.H. IJzerman A.P. (2020), Design and pharmacological profile of a novel covalent partial agonist for the adenosine A1 receptor, Biochemical Pharmacology 180: 114144.
- Yang X., Veldhoven J.P.D. van, Offringa J., Kuiper B.J., Lenselink E.B., Heitman L.H., Es D. van der & IJzerman A.P. (2019), Development of Covalent Ligands for G Protein-Coupled Receptors: A Case for the Human Adenosine A3 Receptor, Journal of Medicinal Chemistry 62(7): 3539-3552.
- Willacey C.C.W., Naaktgeboren M., Moreno E.L., Wegrzyn A.B., Es D. van der, Karu N., Fleming R.M.T., Harms A.C. & Hankemeier T. (2019), LC-MS/MS analysis of the central energy and carbon metabolites in biological samples following derivatization by dimethylaminophenacyl bromide, Journal of Chromatography A 1608: 460413.
- Xia L., Vries H. de, Yang X., Lenselink E.B., Kyrizaki A., Barth F., Louvel J., Dreyer M.K., Es D. van der, IJzerman A.P. & Heitman L.H. (2018), Kinetics of human cannabinoid 1 (CB1) receptor antagonists: Structure-kinetics relationships (SKR) and implications for insurmountable antagonism, Biochemical Pharmacology 151: 166-179.
- Yang X., Michiels T.J.M., Jong C. de, Soethoudt M., Dekker N., Gordon E., Stelt M. van der, Heitman L.H., Es D. van der & IJzerman A.P. (2018), An Affinity-Based Probe for the Human Adenosine A(2A) Receptor, Journal of Medicinal Chemistry 61(17): 7892-7901.
- Es D. van der, Berni F., Hogendorf W.F.J., Meeuwenoord N., Laverde D., Diepen A. van, Overkleeft H.S., Filippov D.V., Hokke C.H., Huebner J., Marel G.A. van der & Codée J.D.C. (2018), Streamlined Synthesis and Evaluation of Teichoic Acid Fragments, Chemistry: a European Journal 24(16): 4014-4018.
- Es D. van der, Hogendorf W.F.J., Overkleeft H.S., Marel G.A. van der & Codee J.D.C. (2017), Teichoic Acids: Synthesis and Applications, Chemical Society Reviews 46: 1464-1482.
- Es D. van der, Groenia N.A., Laverde D., Overkleeft H.S., Huebner J., Marel G.A. van der & Codee J.D.C. (2016), Synthesis of E. faecium wall teichoic acid fragments, Bioorganic & Medicinal Chemistry 24(17): 3893-3907.
- Es D. van der (4 oktober 2016), Synthesis of phosphodiester-containing bacterial cell wall components : teichoic acids, capsular polysaccharides and phosphatidyl glycerol analogues (Dissertatie. Leiden institute of Chemistry (LIC), Science, Leiden University). Promotor(en) en copromotor(en): Marel G.A. van der, Codée J.D.C.