Bert Beerkens
Onderzoeker
- Naam
- Dr. B.L.H. Beerkens
- Telefoon
- +31 71 527 4237
- b.l.h.beerkens@lacdr.leidenuniv.nl
- ORCID iD
- 0000-0002-2884-3961
For more information look at his English website
Onderzoeker
- Wiskunde en Natuurwetenschappen
- Leiden Academic Centre for Drug Research
- LACDR/Medicinal Chemistry
- Beerkens B.L. H., Andrianopoulou V., Wang X., Liu R., Westen G.J. P. van, Jespers W., IJzerman A.P., Heitman L.H. & Es D van der (2024), N-Acyl-N-alkyl sulfonamide probes for ligand-directed covalent labeling of GPCRs: the adenosine A2B receptor as case study, ACS Chemical Biology 19(7): 1554-1562.
- Hollander L.S. den, Beerkens B.L.H., Dekkers S., Veldhoven J.P.D. van, Ortiz Zacarías N.V., Horst C. van der, Sieders E.G., Valk B. de, Wang J., IJzerman A.P., Es D. van der & Heitman L.H (2024), Labeling of CC chemokine receptor 2 with a versatile intracellular allosteric probe, ACS Chemical Biology 19(9): 2070-2080.
- Beerkens B.L.H., Snijders I.M., Snoeck J., Liu R., Tool A.T.J., Le Dévédec S.E., Jespers W., Kuijpers T.W., Westen G.J.P. van, Heitman L.H., IJzerman A.P. & Es D. van der (2023), Development of an affinity-based probe to profile endogenous human adenosine A3 receptor expression, Journal of Medicinal Chemistry 66(16): 11399-11413.
- Beerkens B.L.H. (9 november 2023), Affinity-based profiling of the adenosine receptors (Dissertatie. Leiden Academic Centre for Drug Research (LADCR), Faculty of Science, Leiden University). Promotor(en) en copromotor(en): Ijzerman A.P., Es D. van der.
- Beerkens B.L.H., Wang X., Avgeropoulou M., Adistia L.N., Veldhoven J.P.D. van, Jespers W., Liu R., Heitman L.H., IJzerman A.P. & Es D. van der (2022), Development of subtype-selective covalent ligands for the adenosine A2B receptor by tuning the reactive group, RSC Medicinal Chemistry 13(7): 850-856.
- Beerkens B.L.H., Koc C., Liu R., Florea B.I., Le Dévédec S.E., Heitman L.H., IJzerman A.P. & Es D. van der (2022), A chemical biological approach to study G protein-coupled receptors: labeling the adenosine A1 receptor using an electrophilic covalent probe, ACS Chemical Biology 17(11): 3131-3139.